Amgen Inc.
Synthesis of key intermediate of KRAS G12C inhibitor compound

Last updated:

Abstract:

The present invention relates to an improved, efficient, scalable process to prepare intermediate compounds, such as compound 5M, having the structure ##STR00001## useful for the synthesis of compounds that target KRAS G12C mutations, such as ##STR00002##

Status:
Grant
Type:

Utility

Filling date:

15 Nov 2019

Issue date:

12 Apr 2022