Enanta Pharmaceuticals, Inc.
Process for preparation of sulfonyl carbamate bile acid derivatives

Abstract:

The present invention relates to processes for preparing compounds of Formula (I) and Formula (II): ##STR00001## These compounds are useful as FXR or TGR5 modulators. The present invention also relates to processes for the preparation of the compounds of Formula (III), Formula (IV), Formula (V), and Formula (VI), ##STR00002## The present invention also relates to a process for the preparation of compounds (VII), (VIII) and (IX), ##STR00003##