Takeda Pharmaceutical Company Limited
SOLID STATE FORMS OF FUSED HETEROAROMATIC PYRROLIDINONES

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Abstract:

Disclosed are chemical entities which are inhibitors of spleen tyrosine kinase (SYK), namely, chemical entities comprising 6-((1R,2S)-2-aminocyclohexylamino)-7-fluoro-4-(1-methyl-1H-pyrazol-4-yl)-- 1H-pyrrolo[3,4-c]pyridine-3(2H)-one and certain solid state forms thereof. Also disclosed are methods of using the chemical entities to treat disorders such as a cancer.

Status:
Application
Type:

Utility

Filling date:

8 May 2020

Issue date:

29 Oct 2020