Sale
F2 VISION SCS 10 percent owner 10 percent owner
Common Stock 35,158 $11.23 $394,824 Sale
F2 VISION SCS 10 percent owner 10 percent owner
Common Stock 34,189 $10.48 $358,335 Sale
F2 VISION SCS 10 percent owner 10 percent owner
Common Stock 85,319 $9.96 $850,033 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 17,744 $9.14 $162,091 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 38,558 $9.14 $352,227 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 53,598 $9.14 $489,618 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 457,001 $9.06 $4,140,429 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 542,999 $9.06 $4,919,571 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 9,402 $10.75 $101,072 Purchase
BVF PARTNERS L P/IL 10 percent owner 10 percent owner
Common Stock 266,598 $10.75 $2,865,929 Option
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Stock Option (Right to Buy) 4,000 $4.3 $17,200 Sale
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 400 $23.61 $9,444 Sale
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 204 $22.4 $4,570 Sale
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 3,396 $21.1 $71,656 Option
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 4,000 $4.3 $17,200 Sale
ZAWEL LEIGH officer: Chief Scientific Officer, Small Molec.. officer: Chief Scientific Offic..
Common Stock 19,574 $25 $489,350 Option
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Stock Option (Right to Buy) 8,000 $4.3 $34,400 Sale
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Common Stock 8,000 $25 $200,000 Option
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Common Stock 8,000 $4.3 $34,400 Sale
ZAWEL LEIGH officer: Chief Scientific Officer, Small Molec.. officer: Chief Scientific Offic..
Common Stock 1,079 $25 $26,975 Sale
ZAWEL LEIGH officer: Chief Scientific Officer, Small Molec.. officer: Chief Scientific Offic..
Common Stock 7,468 $25.16 $187,895 Option
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Stock Option (Right to Buy) 4,000 $4.3 $17,200 Sale
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 4,000 $24.77 $99,080 Option
MICHAELSON JENNIFER officer: Chief Development Officer, Bi.. officer: Chief Development Offi..
Common Stock 4,000 $4.3 $17,200 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 3,556 $29.06 $103,337 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 3,124 $29.06 $90,783 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 7,313 $29.16 $213,247 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 6,425 $29.16 $187,353 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 8,088 $29.17 $235,927 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 7,106 $29.17 $207,282 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 4,092 $29.1 $119,077 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 3,595 $29.1 $104,615 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 5,931 $29.04 $172,236 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 6,751 $29.04 $196,049 Sale
UBS ONCOLOGY IMPACT FUND L.P. 10 percent owner 10 percent owner
Common Stock 13,727 $29.35 $402,887 Sale
GADICKE ANSBERT director, 10 percent owner director, 10 percent owner
Common Stock 15,625 $29.35 $458,594 Sale
GADICKE ANSBERT
Common Stock 12,341 $29.11 $359,247 Sale
UBS ONCOLOGY IMPACT FUND L.P.
Common Stock 10,842 $29.11 $315,611 Option
BAEUERLE PATRICK
Common Stock 11,000 $4.3 $47,300 Sale
BAEUERLE PATRICK
Common Stock 11,000 $4.3 $47,300 Option
BAEUERLE PATRICK
Stock Option (Right to Buy) 11,000 $4.3 $47,300 Option
TRIGILIO JEFFREY
Common Stock 15,000 $4.3 $64,500 Sale
TRIGILIO JEFFREY
Common Stock 15,000 $28.34 $425,100 Option
TRIGILIO JEFFREY
Stock Option (Right to Buy) 15,000 $4.3 $64,500 Sale
BAEUERLE PATRICK officer: See Remarks officer: See Remarks
Common Stock 11,000 $4.3 $47,300 Option
BAEUERLE PATRICK officer: See Remarks officer: See Remarks
Common Stock 11,000 $28.45 $312,950 Option
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Common Stock 15,000 $28.34 $425,100 Sale
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Stock Option (Right to Buy) 5,487 $4.3 $23,594 Sale
TRIGILIO JEFFREY officer: Chief Financial Officer officer: Chief Financial Officer
Common Stock 15,000 $4.3 $64,500 Sale
ZAWEL LEIGH
Common Stock 28,118 $28.95 $814,016