Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 45,000 $21.09 $948,870 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 50,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 25,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 62,700 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Call Option (Obligation to sell) 46 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Call Option (Obligation to sell) 157 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Call Option (Obligation to sell) 100 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Call Option (Obligation to sell) 70 $15 $1,050 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 17,100 $5.04 $86,099 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 10,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 261,915 $5 $1,309,575 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 38,085 $5.01 $190,615 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 3,000 $4.91 $14,739 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 35,000 $5.73 $200,655 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 30,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 5,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 35,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 106,000 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 101,010 N/A N/A Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 263,250 $2.18 $574,148 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 6,000 $2 $12,000 Option
BOEHM RAINER J. director director
Stock Option (Right to Buy) 238,625 $0.67 $158,686 Option
SAVAGE ROBERT G. director director
Stock Option (Right to Buy) 100,000 $0.67 $66,500 Option
DURRANT CAMERON director, officer: Chief Executive Officer director, officer: Chief Execut..
Employee Stock Option Exercise (Right to Buy) 75,000 $0.67 $49,875 Option
DURRANT CAMERON director, officer: Chief Executive Officer director, officer: Chief Execut..
Employee Stock Option Exercise (Right to Buy) 75,000 $0.67 $49,875 Purchase
CHAPPELL DALE 10 percent owner, officer: Chief Scientific .. 10 percent owner, officer: Chie..
Common Stock, $0.001 par value 32,028,669 $0.09 $3,010,695 Purchase
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 29,893,424 $0.28 $8,370,159 Sale
NOMIS BAY LTD. 10 percent owner 10 percent owner
Common Stock 38,900 $0.46 $17,894 Sale
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 309,723 $3.1 $960,141 Sale
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 1,913,206 $3.1 $5,930,939 Purchase
HARRISON MICHAEL WAYNE director director
Common Stock 1,705 $29.32 $49,991 Purchase
ANTHION PARTNERS II LLC 10 percent owner 10 percent owner
Common Stock 6,820 $29.32 $199,962 Purchase
BIESTEK MAREK director, other: See Remarks director, other: See Remarks
Common Stock 10,000 $29.32 $293,200 Purchase
FERNANDEZ THOMAS EDWARD director director
Common Stock 6,821 N/A N/A Purchase
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 5,000 $38.15 $190,750 Purchase
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 5,000 $18.88 $94,400 Purchase
BIESTEK MAREK director, other: See Remarks director, other: See Remarks
Common Stock 40,000 $2.04 $81,600 Purchase
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 440,000 $2.02 $888,800 Purchase
ANTHION PARTNERS II LLC 10 percent owner 10 percent owner
Common Stock 150,000 N/A N/A Purchase
ANTHION PARTNERS II LLC 10 percent owner 10 percent owner
Common Stock 113,800 $1.69 $192,322 Purchase
BIESTEK MAREK director, other: See Remarks director, other: See Remarks
Common Stock 135,000 $1.83 $247,050 Purchase
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 613,677 $2.18 $1,337,816 Purchase
ANTHION PARTNERS II LLC 10 percent owner 10 percent owner
Common Stock 243,063 $1.51 $367,025 Purchase
BIESTEK MAREK director, other: See Remarks director, other: See Remarks
Common Stock 65,000 $1.36 $88,400 Purchase
SHKRELI MARTIN 10 percent owner 10 percent owner
Common Stock 597,438 $1.02 $609,387 Purchase
SANOFI other: Former 10% owner other: Former 10% owner
Common Stock 87,500 $8 $700,000 Purchase
HEALY JAMES director director
Common Stock 375,000 $8 $3,000,000 Purchase
SMITH BRIGITTE director director
Common Stock 25,000 $8 $200,000 Purchase
GBS VENTURE PARTNERS PTY, LTD 10 percent owner 10 percent owner
Common Stock 25,000 $8 $200,000 Purchase
5AM PARTNERS LLC 10 percent owner 10 percent owner
Common Stock 62,500 $8 $500,000