| Utility: Co-crystal forms of a novobiocin analog and proline Filling date: 7 Sep 2025 Issue date: 2 Aug 2022 | 5 Jun 2020 | 2 Aug 2022 |
| Utility: PYRIMIDINE TRICYCLIC ENONE DERIVATIVES FOR INHIBITION OF ROR-GAMMA AND OTHER USES Filling date: 7 Sep 2025 Issue date: 5 May 2022 | 18 Jan 2022 | 5 May 2022 |
| Utility: Pyrimidine tricyclic enone derivatives for inhibition of ROR-gamma and other uses Filling date: 7 Sep 2025 Issue date: 5 Apr 2022 | 16 Dec 2017 | 5 Apr 2022 |
| Utility: ANTIOXIDANT INFLAMMATION MODULATORS: OLEANOLIC ACID DERIVATIVES WITH AMINO AND OTHER MODIFICATIONS AT C-17 Filling date: 7 Sep 2025 Issue date: 27 Jan 2022 | 9 Jul 2021 | 27 Jan 2022 |
| Utility: Pyrazolyl and pyrimidinyl tricyclic enones as antioxidant inflammation modulators Filling date: 7 Sep 2025 Issue date: 7 Dec 2021 | 3 Dec 2019 | 7 Dec 2021 |
| Utility: 2,2-DIFLUOROPROPIONAMIDE DERIVATIVES OF BARDOXOLONE METHYL, POLYMORPHIC FORMS AND METHODS OF USE THEREOF Filling date: 7 Sep 2025 Issue date: 18 Nov 2021 | 25 Jun 2021 | 18 Nov 2021 |
| Utility: PYRAZOLE AND IMIDAZOLE COMPOUNDS FOR INHIBITION OF IL-17 AND RORGAMMA Filling date: 7 Sep 2025 Issue date: 23 Sep 2021 | 17 Jun 2019 | 23 Sep 2021 |
| Utility: BIARYL AMIDES WITH MODIFIED SUGAR GROUPS FOR TREATMENT OF DISEASES ASSOCIATED WITH HEAT SHOCK PROTEIN PATHWAY Filling date: 7 Sep 2025 Issue date: 26 Aug 2021 | 14 May 2019 | 26 Aug 2021 |
| Utility: Antioxidant inflammation modulators: oleanolic acid derivatives with amino and other modifications at c-17 Filling date: 7 Sep 2025 Issue date: 17 Aug 2021 | 10 Feb 2020 | 17 Aug 2021 |
| Utility: 2,2-difluoropropionamide derivatives of bardoxolone methyl, polymorphic forms and methods of use thereof Filling date: 7 Sep 2025 Issue date: 3 Aug 2021 | 14 Jun 2017 | 3 Aug 2021 |
| Utility: Imidazolyl tricyclic enones as antioxidant inflammation modulators Filling date: 7 Sep 2025 Issue date: 13 Jul 2021 | 12 Feb 2016 | 13 Jul 2021 |
| Utility: METHODS OF TREATING ALPORT SYNDROME USING BARDOXOLONE METHYL OR ANALOGS THEREOF Filling date: 7 Sep 2025 Issue date: 3 Jun 2021 | 11 Feb 2021 | 3 Jun 2021 |
| Utility: CYSTEINE-DEPENDENT INVERSE AGONISTS OF NUCLEAR RECEPTORS ROR-GAMMA/ROR-GAMMA-T AND METHODS OF TREATING DISEASES OR DISORDERS THEREWITH Filling date: 7 Sep 2025 Issue date: 20 May 2021 | 20 Jun 2019 | 20 May 2021 |
| Utility: C17-HETEROARYL DERIVATIVES OF OLEANOLIC ACID AND METHODS OF USE THEREOF Filling date: 7 Sep 2025 Issue date: 13 May 2021 | 28 Dec 2020 | 13 May 2021 |
| Utility: Methods of treating Alport syndrome using bardoxolone methyl or analogs thereof Filling date: 7 Sep 2025 Issue date: 23 Mar 2021 | 8 Nov 2017 | 23 Mar 2021 |
| Utility: C17 POLAR-SUBSTITUTED HETEROAROMATIC SYNTHETIC TRITERPENOIDS AND METHODS OF USE THEREOF Filling date: 7 Sep 2025 Issue date: 11 Feb 2021 | 20 Jul 2020 | 11 Feb 2021 |
| Utility: C17-heteroaryl derivatives of oleanolic acid and methods of use thereof Filling date: 7 Sep 2025 Issue date: 26 Jan 2021 | 31 Jul 2019 | 26 Jan 2021 |
| Utility: CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE Filling date: 7 Sep 2025 Issue date: 5 Nov 2020 | 5 Jun 2020 | 5 Nov 2020 |
| Utility: ANTIOXIDANT INFLAMMATION MODULATORS: OLEANOLIC ACID DERIVATIVES WITH AMINO AND OTHER MODIFICATIONS AT C-17 Filling date: 7 Sep 2025 Issue date: 30 Jul 2020 | 10 Feb 2020 | 30 Jul 2020 |
| Utility: Co-crystal forms of a novobiocin analog and proline Filling date: 7 Sep 2025 Issue date: 21 Jul 2020 | 1 Feb 2019 | 21 Jul 2020 |
| Utility: PYRAZOLYL AND PYRIMIDINYL TRICYCLIC ENONES AS ANTIOXIDANT INFLAMMATION MODULATORS Filling date: 7 Sep 2025 Issue date: 2 Jul 2020 | 3 Dec 2019 | 2 Jul 2020 |
| Utility: C17-HETEROARYL DERIVATIVES OF OLEANOLIC ACID AND METHODS OF USE THEREOF Filling date: 7 Sep 2025 Issue date: 30 Apr 2020 | 31 Jul 2019 | 30 Apr 2020 |
| Utility: PYRIMIDINE TRICYCLIC ENONE DERIVATIVES FOR INHIBITION OF ROR-GAMMA AND OTHER USES Filling date: 7 Sep 2025 Issue date: 30 Apr 2020 | 16 Dec 2017 | 30 Apr 2020 |
| Utility: Antioxidant inflammation modulators: oleanolic acid derivatives with amino and other modifications at C-17 Filling date: 7 Sep 2025 Issue date: 11 Feb 2020 | 28 Aug 2018 | 11 Feb 2020 |
| Utility: C17-alkanediyl and alkenediyl derivatives of oleanolic acid and methods of use thereof Filling date: 7 Sep 2025 Issue date: 10 Dec 2019 | 15 Feb 2017 | 10 Dec 2019 |
| Utility: METHODS OF TREATING ALPORT SYNDROME USING BARDOXOLONE METHYL OR ANALOGS THEREOF Filling date: 7 Sep 2025 Issue date: 21 Nov 2019 | 8 Nov 2017 | 21 Nov 2019 |
| Utility: C17-heteroaryl derivatives of oleanolic acid and methods of use thereof Filling date: 7 Sep 2025 Issue date: 3 Sep 2019 | 3 Jan 2018 | 3 Sep 2019 |
| Utility: CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE Filling date: 7 Sep 2025 Issue date: 8 Aug 2019 | 1 Feb 2019 | 8 Aug 2019 |