Loxo Oncology
Patents, Design & Utilities

Last updated:

List of all Loxo Oncology patents 37 in total

Status Patent
Application
Utility: FORMULATIONS OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 30 Jun 2022
Application
Utility: METHODS OF DIAGNOSING AND TREATING CANCER External link
Filling date: 5 Sep 2025 Issue date: 24 Mar 2022
Application
Utility: FORMULATIONS OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 24 Mar 2022
Application
Utility: COMPOUNDS USEFUL AS KINASE INHIBITORS External link
Filling date: 5 Sep 2025 Issue date: 3 Mar 2022
Grant
Utility: Process for the preparation of (S)-N-(5-((R)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrim- idin-3-yl)-3-hydroxypyrrolidine-1-carboxamide and salts thereof External link
Filling date: 5 Sep 2025 Issue date: 4 Jan 2022
Application
Utility: PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 9 Dec 2021
Grant
Utility: Methods of treating pediatric cancers External link
Filling date: 5 Sep 2025 Issue date: 7 Dec 2021
Application
Utility: SPRAY-DRIED DISPERSIONS, FORMULATIONS, AND POLYMORPHS OF (S)-5-AMINO-3-(4-((5-FLUORO-2-METHOXYBENZAMIDO)METHYL)PHENYL)-1-(1,1,1-TR- IFLUOROPROPAN-2-YL)-1H-PYRAZOLE-4-CARBOXAMIDE External link
Filling date: 5 Sep 2025 Issue date: 28 Oct 2021
Grant
Utility: Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6- -diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-car- bontrile External link
Filling date: 5 Sep 2025 Issue date: 24 Aug 2021
Grant
Utility: Process for the preparation of pyrazolo[1,5-a]pyrimidines and salts thereof External link
Filling date: 5 Sep 2025 Issue date: 17 Aug 2021
Application
Utility: POINT MUTATIONS IN TRK INHIBITOR-RESISTANT CANCER AND METHODS RELATING TO THE SAME External link
Filling date: 5 Sep 2025 Issue date: 3 Jun 2021
Application
Utility: COMPOUNDS USEFUL AS KINASE INHIBITORS External link
Filling date: 5 Sep 2025 Issue date: 1 Apr 2021
Application
Utility: FORMULATIONS OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 18 Mar 2021
Grant
Utility: Compounds useful as kinase inhibitors External link
Filling date: 5 Sep 2025 Issue date: 16 Feb 2021
Grant
Utility: Point mutations in TRK inhibitor-resistant cancer and methods relating to the same External link
Filling date: 5 Sep 2025 Issue date: 2 Feb 2021
Application
Utility: TREATMENT OF TRK-ASSOCIATED CANCERS External link
Filling date: 5 Sep 2025 Issue date: 28 Jan 2021
Application
Utility: LIQUID FORMULATIONS OF (S)-N-(5-((R)-2-(2,5-DIFLUOROPHENYL)-PYRROLIDIN-1-YL)-PYRAZOLO[1,5-A]PYRI- MIDIN-3-YL)-3-HYDROXYPYRROLIDINE-1-CARBOXAMIDE External link
Filling date: 5 Sep 2025 Issue date: 29 Oct 2020
Application
Utility: PROCESS FOR THE PREPARATION OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 1 Oct 2020
Grant
Utility: Formulations of 6-(2-hydroxy-2-methylpropxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-- diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-A]pyridine-3-carb- onitrile External link
Filling date: 5 Sep 2025 Issue date: 29 Sep 2020
Application
Utility: COMPOUNDS USEFUL AS KINASE INHIBITORS External link
Filling date: 5 Sep 2025 Issue date: 3 Sep 2020
Grant
Utility: Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6- -diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-car- bonitrile External link
Filling date: 5 Sep 2025 Issue date: 18 Aug 2020
Application
Utility: METHODS OF TREATING PEDIATRIC CANCERS External link
Filling date: 5 Sep 2025 Issue date: 30 Jul 2020
Grant
Utility: Point mutations in TRK inhibitor-resistant cancer and methods relating to the same External link
Filling date: 5 Sep 2025 Issue date: 28 Jul 2020
Application
Utility: PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF External link
Filling date: 5 Sep 2025 Issue date: 9 Jul 2020
Grant
Utility: Compounds useful as kinase inhibitors External link
Filling date: 5 Sep 2025 Issue date: 30 Jun 2020
Grant
Utility: Liquid formulations of (S)-N-(5-((R)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyri- midin-3-yl)-3-hydroxypyrrolidine-1-carboxamide External link
Filling date: 5 Sep 2025 Issue date: 2 Jun 2020
Grant
Utility: Point mutations in TRK inhibitor-resistant cancer and methods relating to the same External link
Filling date: 5 Sep 2025 Issue date: 19 May 2020
Grant
Utility: Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer External link
Filling date: 5 Sep 2025 Issue date: 7 Apr 2020
Grant
Utility: Methods of treating pediatric cancers External link
Filling date: 5 Sep 2025 Issue date: 17 Mar 2020
Grant
Utility: Pyrazolopyrimidine derivatives useful as inhibitors of Bruton's tyrosine kinase External link
Filling date: 5 Sep 2025 Issue date: 21 Jan 2020
Grant
Utility: Compounds useful as kinase inhibitors External link
Filling date: 5 Sep 2025 Issue date: 5 Nov 2019
Grant
Utility: Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer External link
Filling date: 5 Sep 2025 Issue date: 3 Sep 2019
Grant
Utility: Pyrazolopyrimidine derivatives as BTK inhibitors for the treatment of cancer External link
Filling date: 5 Sep 2025 Issue date: 3 Sep 2019
Application
Utility: FORMULATIONS OF 6-(2-HYDROXY-2-METHYLPROPOXY)-4-(6-(6-((6-METHOXYPYRIDIN-3-YL)METHYL)-3,6- -DIAZABICYCLO[3.1.1]HEPTAN-3-YL)PYRIDIN-3-YL)PYRAZOLO[1,5-A]PYRIDINE-3-CAR- BONITRILE External link
Filling date: 5 Sep 2025 Issue date: 29 Aug 2019
Application
Utility: FORMULATIONS OF A MACROCYCLIC TRK KINASE INHIBITOR External link
Filling date: 5 Sep 2025 Issue date: 15 Aug 2019
Grant
Utility: Point mutations in TRK inhibitor-resistant cancer and methods relating to the same External link
Filling date: 5 Sep 2025 Issue date: 13 Aug 2019
Grant
Utility: Point mutations in TRK inhibitor-resistant cancer and methods relating to the same External link
Filling date: 5 Sep 2025 Issue date: 6 Aug 2019

Showing 1 to 37 of 37 patents.