Sale
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 1,279,820 $0.66 $845,961 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 250,000 $2.35 $587,500 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Warrants (right to buy) 769,334 $2.35 $1,807,935 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Prefunded Warrants (right to buy) 134,667 $0 $135 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 4,255,319 $0.47 $2,000,000 Option
KIM JASON S. officer: See remarks officer: See remarks
Stock Option (right to buy) 12,089 $0.71 $8,583 Option
KIM JASON S. officer: See remarks officer: See remarks
Common Stock 12,089 $0.71 $8,583 Purchase
MCLENNAN SEAN officer: See remarks officer: See remarks
Common Stock 30,000 $0.82 $24,480 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 200,000 $1.18 $236,200 Option
POMA ERIC E director, officer: See remarks director, officer: See remarks
Stock Option (right to buy) 27,325 $0.71 $19,401 Option
POMA ERIC E director, officer: See remarks director, officer: See remarks
Common Stock 27,325 $0.71 $19,401 Option
POMA ERIC E director, officer: See remarks director, officer: See remarks
Common Stock 6,831 $0.71 $4,850 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 200,000 $4.04 $807,200 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 750,000 $6 $4,500,000 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 100,000 $6.13 $613,000 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 75,000 $7.09 $531,825 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $7 $559,840 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 125,000 $7.13 $891,625 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 119,382 $6.96 $830,779 Option
POMA ERIC E director, officer: See remarks director, officer: See remarks
Common Stock 3,563 N/A N/A Option
POMA ERIC E director, officer: See remarks director, officer: See remarks
Stock Option (right to buy) 3,563 N/A N/A Option
KIM JASON S. officer: See remarks officer: See remarks
Common Stock 32,038 $0.71 $22,747 Sale
KIM JASON S. officer: See remarks officer: See remarks
Common Stock 2,770 $8.36 $23,157 Option
KIM JASON S. officer: See remarks officer: See remarks
Stock Option (right to buy) 32,038 $0.71 $22,747 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 40,852 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 150,000 $8.62 $1,292,700 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 150,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 100,000 $7.81 $781,000 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 50,000 $8.02 $400,850 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 235,664 $8.23 $1,939,750 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 300,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 200,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 200,000 $9.44 $1,887,200 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $11.45 $915,840 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 75,000 $11.48 $860,850 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 235,004 $11.29 $2,652,960 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 1,185,770 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $11.69 $935,360 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $11.94 $955,040 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 320,000 $8.29 $2,651,840 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 320,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 125,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $9.16 $732,480 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 N/A N/A Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 470,335 $8.33 $3,919,772 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 75,000 $10.86 $814,200 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $8.83 $706,320 Purchase
BIOTECH TARGET N V 10 percent owner 10 percent owner
Common Stock 80,000 $8.83 $706,320 Sale
SHV MANAGEMENT SERVICES, LLC 10 percent owner 10 percent owner
Common Stock 500,000 $13.05 $6,525,000 Sale
LALANDE KEVIN M. director, 10 percent owner director, 10 percent owner
Common Stock 500,000 $13.05 $6,525,000