Sale
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Common Stock 91,898 $21.01 $1,930,317 Option
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Stock Option (Right to Buy) 13,978 N/A N/A Sale
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Common Stock 23,650 $21.4 $506,157 Option
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Common Stock 23,650 $4.16 $98,337 Sale
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Common Stock 13,978 $21.95 $306,803 Option
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Common Stock 13,978 $21.95 $306,803 Option
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Stock Option (Right to Buy) 8,297 $2.55 $21,157 Option
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Stock Option (Right to Buy) 5,800 $2.55 $14,790 Option
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Common Stock 5,800 $22.68 $131,515 Sale
ZORN PETER A officer: SVP, Lgl Affrs, GC & Secretary officer: SVP, Lgl Affrs, GC & S..
Common Stock 5,800 $22.68 $131,515 Option
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Stock Option (Right to Buy) 5,800 $1.75 $10,150 Sale
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Common Stock 5,800 $1.75 $10,150 Option
BRENNAN JEFFREY P officer: SVP, Bus. and Comm. Dev. & CBO officer: SVP, Bus. and Comm. De..
Common Stock 5,800 $1.75 $10,150 Sale
BVF PARTNERS L P/IL other: See Explanation of Responses other: See Explanation of Respo..
Common Stock 638,400 $23.6 $15,063,048 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 11,000 $1.75 $19,250 Sale
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 11,000 $1.75 $19,250 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Stock Option (Right to Buy) 11,000 $1.75 $19,250 Sale
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 9,050 $16.27 $147,225 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Stock Option (Right to Buy) 9,050 $16.27 $147,225 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 9,050 $16.27 $147,225 Sale
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 950 $1.75 $1,663 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 950 $1.75 $1,663 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Stock Option (Right to Buy) 950 $1.75 $1,663 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Stock Option (Right to Buy) 851 $15 $12,765 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 851 $15 $12,765 Sale
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 851 $15 $12,765 Sale
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 10,000 $1.75 $17,500 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 11,149 $1.75 $19,511 Sale
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Common Stock 2,100 $1.75 $3,675 Option
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Common Stock 2,100 $1.75 $3,675 Sale
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 11,149 $1.75 $19,511 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Common Stock 10,000 $1.75 $17,500 Option
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Stock Option (Right to Buy) 8,000 $1.75 $14,000 Option
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Stock Option (Right to Buy) 2,100 $1.75 $3,675 Sale
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Common Stock 8,000 $1.75 $14,000 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Stock Option (Right to Buy) 11,149 $1.75 $19,511 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Stock Option (Right to Buy) 10,000 $1.75 $17,500 Option
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Common Stock 8,000 $1.75 $14,000 Option
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Stock Option (Right to Buy) 13,955 $1.75 $24,421 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Stock Option (Right to Buy) 9,400 $14.54 $136,648 Sale
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Common Stock 5,400 $14.5 $78,300 Option
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Common Stock 13,955 $1.75 $24,421 Sale
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 9,400 $14.54 $136,648 Option
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Common Stock 5,400 $14.5 $78,300 Option
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Stock Option (RIght to Buy) 5,400 $14.5 $78,300 Option
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 9,400 $14.54 $136,648 Sale
CALDWELL WILLIAM S officer: SVP - Drug Discovery and Dev. officer: SVP - Drug Discovery a..
Common Stock 13,955 $1.75 $24,421 Sale
DEBETHIZY J DONALD director, officer: President and CEO director, officer: President an..
Common Stock 600 $1.75 $1,050 Option
DUNBAR GEOFFREY C officer: SVP, Clin. Dev. & Reg. Affairs officer: SVP, Clin. Dev. & Reg...
Stock Option (Right to Buy) 7,900 $14.04 $110,900 Option
MUSSO ALAN A officer: SVP, Fin+Admin, CFO & Treas officer: SVP, Fin+Admin, CFO & ..
Stock Option (Right to Buy) 600 $1.75 $1,050