Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 19,670 $14.86 $292,277 Sale
BAKER BROS. CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 3,535 $14.8 $52,318 Sale
BAKER BIOTECH CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 18,449 $14.8 $273,045 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 1,136 $14.8 $16,813 Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 36,880 N/A N/A Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 17,149 $15.24 $261,368 Sale
BAKER BROS. CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 1,645 $15.24 $25,071 Sale
BAKER BIOTECH CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 8,579 $15.24 $130,753 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 527 $15.24 $8,032 Option
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Stock Options 18,769 N/A N/A Option
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Common Stock 18,769 $4 $75,076 Sale
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Common Stock 7,986 $13.67 $109,153 Sale
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Common Stock 27,600 $13.11 $361,781 Option
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Stock Options 63,784 $2 $127,568 Option
AGRAWAL SUDHIR director, officer: President of Research director, officer: President of..
Common Stock 63,784 $4 $255,136 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 302 $14.51 $4,383 Sale
BAKER BROS. CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 943 $14.51 $13,687 Sale
BAKER BIOTECH CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 4,920 $14.51 $71,409 Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 9,835 $14.51 $142,745 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 776 $14.99 $11,635 Sale
BAKER BIOTECH CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 12,606 $14.99 $189,002 Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 25,202 $14.99 $377,854 Sale
BAKER BROS. CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 2,416 $14.99 $36,223 Sale
BAKER BROS. CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 31,791 $15.41 $489,899 Sale
BAKER BIOTECH CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 165,874 $15.41 $2,556,118 Sale
BAKER BROTHERS LIFE SCIENCES CAPITAL (GP), LLC 10 percent .. 10 percent owner
Common Stock 331,598 $15.41 $5,109,925 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 10,207 $15.41 $157,290 Sale
WYNGAARDEN JAMES B director director
Common Stock 1,284 $14.5 $18,618 Option
WYNGAARDEN JAMES B director director
Warrant to purchase 1,284 $8 $10,272 Option
WYNGAARDEN JAMES B director director
Common Stock 1,284 $8 $10,272 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock Warrants (right to buy) 73,463 $8 $587,704 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock 279,727 $8 $2,237,816 Option
WYNGAARDEN JAMES B director director
Stock Options 4,990 $4 $19,960 Option
WYNGAARDEN JAMES B director director
Common Stock 5,990 $9.4 $56,276 Sale
WYNGAARDEN JAMES B director director
Common Stock 4,990 $4 $19,960 Sale
SULLIVAN TIMOTHY M officer: VP Development Programs officer: VP Development Programs
Common Stock 4,200 $14.95 $62,790 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock 69,202 $5.36 $370,923 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock Warrants (right to buy) 69,202 $5.36 $370,923 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock Warrants (right to buy) 54,065 $5.36 $289,788 Option
WYNGAARDEN JAMES B director director
Common Stock 10,306 $10.04 $103,472 Option
WYNGAARDEN JAMES B director director
Stock Options 10,306 $10.04 $103,472 Option
BEXON ALICE officer: V.P. Clinical Development officer: V.P. Clinical Developm..
Common Stock 27,499 $7.55 $207,617 Sale
WYNGAARDEN JAMES B director director
Common Stock 10,306 $10.04 $103,472 Sale
BEXON ALICE officer: V.P. Clinical Development officer: V.P. Clinical Developm..
Common Stock 27,499 $7.55 $207,617 Option
BEXON ALICE officer: V.P. Clinical Development officer: V.P. Clinical Developm..
Stock Option 27,499 $7.55 $207,617 Option
ZEIN YOUSSEF EL 10 percent owner 10 percent owner
Common Stock 54,065 $5.36 $289,788 Option
WYNGAARDEN JAMES B director director
Common Stock 9,704 $10 $97,040 Sale
WYNGAARDEN JAMES B director director
Common Stock 9,704 $10 $97,040 Option
WYNGAARDEN JAMES B director director
Stock Options 9,704 $2 $19,408 Sale
14159 CAPITAL (GP), LLC 10 percent owner 10 percent owner
Common Stock 13 $13 $169